@article{oai:tohoku-mpu.repo.nii.ac.jp:00000138, author = {渡邉, 一弘 and Watanabe, Kazuhiro and 佐藤, 健志 and Sato, Takeshi and 藤田, 礼子 and Fujita, Reiko}, issue = {54}, journal = {東北薬科大学研究誌, Journal of Tohoku Pharmaceutical University}, month = {Dec}, note = {1-Protected 2(1H)-pyridones are highly useful dienophiles because Diels-Alder reaction of 1-sulfonyl-2(1H)-pyridones gave the synthetic intermediate such as quinoline and isoquinoline derivatives. Acylation of 2(1H)-pyridone bearing a methoxycarbonyl group at the 5 or 6-position with benzoyl chloride having a some functional group (such as bromo, methoxy, nitro) gave 1-benzoylated 2(1H)-pyridone derivatives. Further, the sulfonylation of 3-cyano- and 3-methoxycarbonyl-1(2H)-isoquinolones afforded 2-sulfonylisoquinolone derivative.}, pages = {19--25}, title = {窒素原子上に電子吸引性基を有する2-ピリドン誘導体の合成}, year = {2007}, yomi = {ワタナベ, カズヒロ and サトウ, タケシ and フジタ, レイコ} }